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Oncology Drugs A to Z: FDA Status, Uses & Safety
Browse oncology drugs A to Z with FDA status, approved-use context, safety information, cancer treatment resources, and primary-source links.
Browse oncology drug and regimen pages
Each linked entry has its own crawlable, self-canonical reference page. FDA status and indications can change, so current primary sources are linked whenever a page has been editorially reviewed.
Featured FDA-reviewed oncology drug pages
- Pepaxto (Melphalan flufenamide) — U.S. approval withdrawn
- Revuforj (Revumenib) — FDA approved for specified biomarker-defined acute leukemias
- Avmapki Fakzynja Co-Pack (Avutometinib and defactinib) — FDA accelerated approval for a specified KRAS-mutated ovarian cancer setting
- Lifyorli (Relacorilant) — FDA approved in March 2026 for a specified platinum-resistant cancer setting
- Zepzelca (Lurbinectedin) — FDA approved for specified small-cell lung cancer settings
- Datroway (Datopotamab deruxtecan-dlnk) — FDA approved for specified breast and lung cancer settings
A
- ABVD
- AC
- Abemaciclib (Verzenios)
- Abiraterone (Zytiga)
- Abraxane
- Abstral
- Acalabrutinib (Calquence)
- Actimorph
- Actinomycin D
- Actiq
- Adriamycin
- Afatinib (Giotrif)
- Afinitor
- Aflibercept and folinic acid, fluorouracil and irinotecan (FOLFIRI)
- Aldara
- Alectinib (Alecensa)
- Alpelisib and fulvestrant
- Anastrozole (Arimidex)
- Apalutamide
- Ara C
- Arimidex
- Aromasin
- Arsenic trioxide and tretinoin
- Asciminib (Scemblix)
- Asparaginase (Spectrila, Erwinase, Oncaspar)
- Atezolizumab (Tecentriq)
- Atezolizumab and bevacizumab
- Atezolizumab and nab-paclitaxel
- Avelumab (Bavencio)
- Adagrasib (Krazati)
- Afamitresgene autoleucel (Tecelra)
- Amivantamab and hyaluronidase-lpuj (Rybrevant Faspro)
- Avapritinib (Ayvakit)
- Avutometinib and defactinib (Avmapki Fakzynja co-pack)
- Axatilimab-csfr (Niktimvo)
- Axicabtagene ciloleucel (Yescarta)
- Axitinib (Inlyta)
- Azacitidine (Vidaza)
- Azacitidine tablets (Onureg)
B
- BEACOPDac
- BEACOPP
- BEAM
- Belzutifan (Welireg)
- Bendamustine (Levact)
- Besponsa
- Bevacizumab (Avastin)
- Bexarotene (Targretin)
- Bicalutamide (Casodex)
- Bleomycin
- Bleomycin, etoposide and platinum (BEP)
- Belantamab mafodotin-blmf (Blenrep)
- Belumosudil (Rezurock)
- Blinatumomab (Blincyto)
- Brexucabtagene autoleucel (Tecartus)
- Bortezomib (Velcade)
- Bortezomib, cyclophosphamide and dexamethasone (VCD)
- Bosulif
- Bosutinib (Bosulif)
- Brentuximab
- Brigatinib
- Buserelin (Suprefact or Suprecur)
- Busulfan
C
- CAPOX
- CAPTEM
- CAV chemotherapy
- CCNU
- CHOP
- CPX351
- Cabazitaxel
- Cabometyx
- Cabozantinib capsules (Cometriq)
- Cabozantinib tablets (Cabometyx)
- Capmatinib (Tabrecta)
- Caelyx
- Ciltacabtagene autoleucel (Carvykti)
- Cosibelimab-ipdl (Unloxcyt)
- Campto
- Capecitabine
- Capecitabine and temozolomide (CAPTEM)
- Capivasertib and fulvestrant
- CarboTaxol
- Carboplatin
- Carboplatin and etoposide
- Carboplatin and paclitaxel
- Carfilzomib and dexamethasone
- Casodex
- Cemiplimab (Libtayo)
- Ceritinib (Zykadia)
- Cetuximab (Erbitux)
- Chlorambucil
- Cisplatin
- Cisplatin and capecitabine (CX)
- Cisplatin and fluorouracil (5FU)
- Cisplatin, etoposide and ifosfamide (VIP)
- Cisplatin, fluorouracil (5FU) and trastuzumab
- Cladribine
- Columvi
- Cometriq
- Crizotinib (Xalkori)
- Cyclophosphamide
- Cyclophosphamide, thalidomide and dexamethasone (CTD)
- Cyprostat
- Cyproterone acetate (Cyprostat)
- Cytarabine (Ara C, cytosine arabinoside)
- Cytarabine into spinal fluid (intrathecal cytarabine)
- Cytosine arabinoside
D
- DA
- DHAP
- DTIC
- Dabrafenib (Tafinlar)
- Dabrafenib and trametinib
- Dacarbazine
- Dacomitinib (Vizimpro)
- Dactinomycin (actinomycin D)
- Daratumumab
- Daratumumab, bortezomib, thalidomide and dexamethasone (DVTD)
- Daratumumab, lenalidomide and dexamethasone (DRD)
- Darolutamide (Nubeqa)
- Darzalex
- Dasatinib
- Daunorubicin and cytarabine (DA)
- Daunorubicin, cytarabine and midostaurin
- Decapeptyl SR (breast cancer)
- Degarelix (Firmagon)
- Denosumab injection (Prolia, Xgeva)
- Dexamethasone
- Diamorphine
- Docetaxel (Taxotere)
- Docetaxel and nintedanib
- Datopotamab deruxtecan-dlnk (Datroway)
- Decitabine and cedazuridine (Inqovi)
- Docetaxel, cisplatin and fluorouracil (TPF)
- Dordaviprone (Modeyso)
- Dostarlimab (Jemperli)
- Doxorubicin
- Doxorubicin and ifosfamide
- Durogesic
- Durvalumab (Imfinzi)
E
- EC
- ECF
- EOX
- EP
- ESHAP
- Effentora
- Eflornithine (Iwilfin)
- Elacestrant (Korserdu)
- Elranatamab-bcmm (Elrexfio)
- Encorafenib and binimetinib
- Enfortumab vedotin-ejfv (Padcev)
- Ensartinib (Ensacove)
- Erdafitinib (Balversa)
- Encorafenib and cetuximab
- Entrectinib (Rozlytrek)
- Enzalutamide (Xtandi)
- Epcoritamab (Tepkinly)
- Epirubicin (Pharmorubicin)
- Epirubicin, cisplatin and capecitabine (ECX)
- Epirubicin, oxaliplatin and fluorouracil (EOF)
- Erbitux
- Eribulin (Halaven)
- Erlotinib (Tarceva)
- Erwinase
- Etopophos
- Etoposide (Etopophos)
- Etoposide and Cisplatin (EP)
- Everolimus (Afinitor)
- Exemestane (Aromasin)
F
- FLAG
- FLAG-Ida
- FLOT
- FOLFIRINOX
- FOLFOX
- FOLFOXIRI
- Faslodex
- Femara
- Fentanyl
- Firmagon
- Fludara
- Fludarabine
- Fludarabine, cyclophosphamide and rituximab (FCR)
- Fluorouracil (5FU)
- Fluorouracil, leucovorin, oxaliplatin and docetaxel (FLOT)
- Flutamide
- Folinic acid, fluorouracil and irinotecan (FOLFIRI)
- Folinic acid, fluorouracil and oxaliplatin (FOLFOX)
- Folinic acid, fluorouracil, oxaliplatin and irinotecan (FOLFOXIRI)
- Fotivda
- Fruquintinib (Fruzaqla)
- Fulvestrant (Faslodex)
- Futibatinib (Lytgobi)
G
- G-CSF
- GDP
- Gefitinib (Iressa)
- GemCarbo (gemcitabine and carboplatin)
- GemTaxol
- Gemcitabine
- Gemcitabine and capecitabine (GemCap)
- Gemcitabine and cisplatin (GC)
- Gemcitabine intravesical system (Inlexzo)
- Gemcitabine and nab-paclitaxel
- Gemcitabine and paclitaxel (GemTaxol)
- Gemtuzumab ozogamicin, daunorubicin and cytarabine
- Gemzar
- Gilteritinib (Xospata)
- Giotrif
- Gliadel (carmustine wafers)
- Glivec
- Glofitamab (Columvi)
- Gonapeptyl
- Goserelin for breast cancer
- Goserelin for prostate cancer
- Granulocyte colony stimulating factor (G-CSF)
H
I
- ICE
- IPE
- Ibandronic acid (Bondronat)
- Ibrance
- Ibrutinib (Imbruvica)
- Idarubicin
- Ifosfamide
- Imatinib (Glivec)
- Idecabtagene vicleucel (Abecma)
- Imetelstat (Rytelo)
- Imlunestrant (Inluriyo)
- Inavolisib (Itovebi)
- Irinotecan liposome (Onivyde)
- Isatuximab-irfc (Sarclisa)
- Imiquimod cream (Aldara)
- Inotuzumab ozogamicin (Besponsa)
- Ipilimumab (Yervoy)
- Ipilimumab and nivolumab
- IrCap
- Iressa
- Irinotecan
- Irinotecan and capecitabine (XELIRI, CAPIRI, Ir-Cap, I-Cap)
- Irinotecan de Gramont
- Irinotecan modified de Gramont
- Ivosidenib (Tibsovo)
- Ivosidenib and azacitidine
- Ixazomib, lenalidomide and dexamethasone
J
K
L
- L-DA
- LITAK
- Lanreotide (Somatuline)
- Larotrectinib (Vitrakvi)
- Lenalidomide (Revlimid)
- Lenvatinib (Lenvima, Kisplyx)
- Letrozole (Femara)
- Leuprorelin
- Leustat
- Levact
- Liposomal daunorubicin and cytarabine (Vyxeos, CPX351, L-DA)
- Lomustine
- Loncastuximab tesirine (Zynlonta)
- Lazertinib (Lazcluze)
- Lifileucel (Amtagvi)
- Linvoseltamab-gcpt (Lynozyfic)
- Lisocabtagene maraleucel (Breyanzi)
- Lurbinectedin (Zepzelca)
- Luspatercept-aamt (Reblozyl)
- Lutetium Lu 177 dotatate (Lutathera)
- Lutetium Lu 177 vipivotide tetraxetan (Pluvicto)
- Lonsurf
- Lorlatinib (Lorviqua)
- Lynparza
- Lysodren
- Lytgobi
M
- MAP
- MMM
- MST Continus
- MVAC
- MXL
- Mabthera
- Medroxyprogesterone acetate (Provera)
- Megace
- Megestrol acetate (Megace)
- Margetuximab-cmkb (Margenza)
- Melphalan
- Melphalan flufenamide (Pepaxto)
- Mepact
- Mercaptopurine
- Methotrexate
- Methotrexate, cytarabine, thiotepa and rituximab (MATRix)
- Methylprednisolone
- Midostaurin (Rydapt)
- Midostaurin, daunorubicin and cytarabine
- Mifamurtide (Mepact)
- Mitomycin
- Mirdametinib (Gomekli)
- Mirvetuximab soravtansine-gynx (Elahere)
- Mitomycin intravesical solution (Zusduri)
- Mosunetuzumab-axgb (Lunsumio)
- Mitotane (Lysodren)
- Mitoxantrone
- Mobocertinib (Exkivity)
- Modified de Gramont
- Morphgesic SR
- Morphine (Oramorph, Sevredol, Zomorph, Actimorph)
N
- Nadofaragene firadenovec-vncg (Adstiladrin)
- Nab-paclitaxel (Abraxane)
- Naxitamab (Danyelza)
- Navelbine
- Nelarabine (Atriance)
- Neratinib (Nerlynx)
- Nerlynx
- Nilotinib (Tasigna)
- Nipent
- Nirogacestat (Ogsiveo)
- Niraparib (Zejula)
- Nogapendekin alfa inbakicept-pmln (Anktiva)
- Niraparib and abiraterone acetate (Akeega)
- Nivolumab (Opdivo)
- Nivolumab and relatlimab (Opdualag)
O
P
- PC
- PE
- Paclitaxel
- Paclitaxel and carboplatin (PC, CarboTaxol)
- Palbociclib (Ibrance)
- Pamidronate disodium
- Panitumumab
- Panobinostat, bortezomib and dexamethasone
- Pazopanib (Votrient)
- Peginterferon alfa 2a
- Pegylated liposomal doxorubicin
- Pembrolizumab (Keytruda)
- Pemetrexed (Alimta)
- Pemetrexed and carboplatin
- Pemetrexed and cisplatin
- Pemigatinib (Pemazyre)
- Pentostatin (Nipent)
- Penpulimab-kcqx
- Pirtobrutinib (Jaypirca)
- Pralsetinib (Gavreto)
- Perjeta
- Pertuzumab-dpzb (Poherdy)
- Pertuzumab (Perjeta)
- Phesgo or trastuzumab and pertuzumab
- Polatuzumab vedotin with R-CHP (Pola-R-CHP)
- Polatuzumab vedotin, bendamustine and rituximab (Pola-BR)
- Pomalidomide and dexamethasone
- Ponatinib (Incyte)
- Prednisolone
- Procarbazine
- Procarbazine, lomustine and vincristine (PCV)
- Prolia
- Prostap
- Provera
Q
R
- R-CHOP
- R-CVP
- R-DHAP
- R-ESHAP
- R-GCVP
- R-GDP
- R-Idelalisib
- RICE
- Raloxifene
- Raltitrexed (Tomudex)
- Regorafenib
- Relacorilant (Lifyorli)
- Relugolix (Orgovyx)
- Remestemcel-L-rknd (Ryoncil)
- Repotrectinib (Augtyro)
- Revlimid
- Ripretinib (Qinlock)
- Ribociclib (Kisqali)
- Risedronate sodium
- Retifanlimab-dlwr (Zynyz)
- Rituximab
- Rituximab and idelalisib (R-Idelalisib)
- Rixathon
- Revumenib (Revuforj)
- Rubraca
- Rucaparib (Rubraca)
- Ruxience
- Ruxolitinib (Jakavi)
S
- Sacituzumab govitecan (Trodelvy)
- Selumetinib (Koselugo)
- Selinexor, bortezomib and dexamethasone (SVd)
- Selpercatinib (Retsevmo)
- Sevabertinib (Hyrnuo)
- Sevredol
- Sodium clodronate
- Sorafenib
- Sirolimus protein-bound particles (Fyarro)
- Sotorasib (Lumykras)
- Steroids (dexamethasone, prednisolone, methylprednisolone and hydrocortisone)
- Stivarga
- Streptozocin (Zanosar)
- Sunvozertinib (Zegfrovy)
- Sunitinib (Sutent)
- Sutent
T
- TC
- TIP
- Tafinlar
- Tagrisso
- Talazoparib (Talzenna)
- Talimogene laherparepvec (T-VEC)
- Tamoxifen
- Tarceva
- Targretin
- Tasigna
- Taxol
- Taxotere
- Tafasitamab-cxix (Monjuvi)
- Taletrectinib (Ibtrozi)
- Talquetamab-tgvs (Talvey)
- Tarlatamab-dlle (Imdelltra)
- Tazemetostat (Tazverik)
- Taxotere and cyclophosphamide (TC protocol)
- Tebentafusp (Kimmtrak)
- Tecentriq
- Teclistamab (Tecvayli)
- Telisotuzumab vedotin-tllv (Emrelis)
- Tisagenlecleucel (Kymriah)
- Tisotumab vedotin-tftv (Tivdak)
- Toripalimab-tpzi (Loqtorz)
- Tovorafenib (Ojemda)
- Tremelimumab (Imjudo)
- Temodal
- Temozolomide (Temodal)
- Tepotinib (Tepmetko)
- Thiotepa
- Tivozanib (Fotivda)
- Tomudex
- Topotecan (Hycamtin)
- Trabectedin (Yondelis)
- Trametinib (Mekinist)
- Trastuzumab
- Trastuzumab and pertuzumab
- Trastuzumab deruxtecan (Enhertu)
- Trastuzumab emtansine (Kadcyla)
- Treosulfan (Trecondi)
- Trifluridine and tipiracil (Lonsurf)
- Triptorelin (Decapeptyl SR or Gonapeptyl) for prostate cancer
- Truxima
- Tucatinib, trastuzumab and capecitabine
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